pharm---misc
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- Which ones block cell wall synthesis by inhibiting peptidoglycan cross linking?
-
Penicillin
Ampicillin
Ticarcillin
Piperacillin
Imipenem
Aztreonam
Cephalosporins - Which ones block peptidoglycan synthesis?
-
bacitracin
Vancomycin
Cycloserine - Which ones block protein synthesis at 50S ribosomal subunit?
-
Chloramphenicol
Erythromycin/macrolides
Lincomycin
Clindamycin
Streptogramins(quinupristin, dalfopristin)
Linezolid - Which block protein syntheis at 30S ribosomal subunit?
-
Aminoglycosides
tetracyclines - which ones block nucleotide synthesis?
-
sulfonamides
trimethoprim - block DNA topoisomerases
- Quinolones
- Block mRNA synthesis
- Rifampin
- Bacteriacidal antibiotics
-
Penicillin
cephalosporins
vancomycin
aminoglycosides
fluoroquinolones
metronidazole - disrupt bacterial/fungal cell membranes
- Polymyxins
- disrupt fungal cell membranes
-
Amphotericin B
nystatin
fluconazoles/azoles - Unknown
- Pentamidine
- Ivermectin
- Onchocerciasis (rIVER blindness treated with IVERmectim)
- mebendazole/thiabendazole
- Nematode/roundworm (pinworm, whipworm) infection
- Pyrantel pamote
-
Giant roundworm (ascarias)
Hookworm (
Pinworm - Prazinquantel
-
trematode fluke---(schistosomes, paragonimus, Clonorchis)
cysticercosis - Niclosamide
- Cestode/tapeworm (diphyllobothrium latum, Taenia species) infections not including cysticercosis
- Pentavalent antimony
- Leishmaniasis
- Chloroquine, quinine, mefloquine, atovaquone, proguanil
- Malaria
- Primaquine
- Latent hypnozite (liver) forms of malaria (P vivax, ovale)
- metronidazole
-
Giardiasis
Amoebic dysentary (Entamoeba histolytica)
bacterial vaginitis (gardnerella vaginalis)
Trichomonas - Pentamindine
- P. Carini pneumonia prophylaxis
- Nifurtimox
-
Chagas
American trypanosomiasis (T. cruzi) - Suramin
- African trypanosomiasis (sleeping sickness)