FA Pharmacology: ANS Drugs
Terms
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- Epineprhine: Selectivity and Clinical Application?
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cathecholamine
direct general agonist(a1,a2,B1,B2)
anaphylaxis, glaucoma (open angle), asthma, hypotension - Norepinephrine: Selectivity and Clinical Application?
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catecholamine
a1, a2, B1
Hypotension, (but decreases renal perfusion) - Isoproterenol: Selectivity and Clinical Application?
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catecholamine
B1 = B2
AV block(rare) - Dopamine: Selectivity and Clinical Application?
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catecholamine
D1=D2 >B >a
Shock (increases renal perfusion), heart failure - Dobutamine: Selectivity and Clinical Application?
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catecholamine
B1 >B2
shock, heart failure - Amphetamine: mechanism and clinical application?
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indirect general agonist, release stored catecholamines
Narcolepsy, obesity, ADHD - Ephedrine: mechanism and clinical application?
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indirect general agonist, releases stored catecholamines
nasal decongestant, urinary incontinence, hypotension - Phenylephrine: selectivity and clinical application?
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a1 >a2
pupil dilator, vasonconstriction, nasal decongestion -
Albuterol
Terbutaline
...selectivity and clinical application? -
B2>B1
asthma - Cocaine: mechanism and clinical application?
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indirect general agonist; uptake inhibitor
causes vasoconstriction and local anesthesia - Clonidine: mechanism and clinical application?
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Centrally acting a-agonist, decreases central adrenergic flow
Hypertension, especially with renal disease (no decrease in blood flow to the kidney)